1、BET-IN-4Cat. No.: HY-111916CAS No.: 1801503-93-4Molecular Formula: CHNOMolecular Weight: 375.42Target: Epigenetic Reader DomainPathway: EpigeneticsStorage: Please store the product under the recommended conditions in the COA.BIOLOGICAL ACTIVITYDescription BET-IN-4 is a potent BET bromodomain protein
2、 (BRD4) inhibitor, with an IC50 of 1 M1.IC & Target BRD4 1 M (IC50)In Vitro BET-IN-4 (Compound 50) is a potent BET bromodomain protein (BRD4) inhibitor, with an IC50 of 1 M1.REFERENCES1. Susanta Samajdar, et al. Bicyclic heterocyclic derivatives as bromodomain inhibitors. WO2015104653A1Caution: Product has not been fully validated for medical applications. For research use only.Tel: 609-228-6898 Fax: 609-228-5909 E-mail: techMedChemEAddress: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USAProduct Data Sheet InhibitorsAgonistsScreening Librarieswww.MedChemE1