1、鼀嘁堀吀渀琀攀爀氀攀甀欀椀渀刀攀氀愀琀攀搀渀栀椀戀椀琀漀爀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀攀挀攀昀愀愀搀挀戀攀攀愀愀愀戀挀戀愀攀攀搀昀愀攀脀Vigabatrin-(-Vinyl-GABA)-GABA-Receptor-Inhibitor-MedChemExpress.pdfde9864f4ef52666c8098efc44d42f04429f4e339e93159046cb70e822482e8a00$褀嘁椀猀琀甀猀攀爀琀椀戀娀洀吀伀刀渀栀椀戀椀琀漀爀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀挀搀挀挀愀戀搀昀戀愀攀挀愀攀挀挀愀戀挀搀愀昀茀Vonoprazan-Fumarate-(TAK-438)-Proton-
2、Pump-Inhibitor-MedChemExpress.pdf170d39ce8bd20da386880d58dc9a65b658d74f9a69d6f3fc68abeff11d6a29260$嘁漀爀琀椀漀砀攀琀椀渀攀甀吀刀攀挀攀瀀琀漀爀渀栀椀戀椀琀漀爀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀挀搀戀挀搀搀愀戀搀昀戀戀昀攀攀搀戀挀攀戀搀戀愀攀戀昀攀搀搀蔀Vortioxetine-hydrobromide-(Lu-AA21004-hydrobromide)-5-HT-Receptor-Inhibitor-MedChemExpress.pdf98d3702ae899b9c0a2c7fd371376afc61
3、e0629d219969481b06da5ba532325010$焀嘀唀洀氀甀刀最漀渀椀猀琀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀挀搀挀昀挀搀搀昀挀昀戀挀戀搀愀昀挀搀昀昀搀攀戀攀挀挀愀挀攀戀蜀qVU-0364439-mGluR-Agonist-MedChemExpress.pdf4334bdaa962da9ad58c792f876106d175031ef8a3746e7f6291d740f98529c070$洀圀夀洀吀伀刀渀栀椀戀椀琀漀爀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀攀攀搀愀愀愀昀攀愀搀戀搀戀攀攀搀搀昀搀攀戀愀搀攀褀WAY-163909-5-HT-Receptor-Agonist-MedChemExpre
4、ss.pdfffc394026608ed54be59fccb65a37718f66258442a8bb2c47c9130386acb144a0$欀圀倀匀吀吀渀栀椀戀椀琀漀爀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀昀愀昀搀愀愀戀愀愀昀搀戀搀昀戀昀戀攀戀戀挀戀愀攀攀戀謀(R)-(-)-Gossypol-(AT-101)-Bcl-2-Family-Inhibitor-MedChemExpress.pdf22366af51de0a475b8703ed4b39bdde8532b29c2d9d8b14c79cae9d2a5be4bfe0唁刀漀猀猀礀瀀漀氀愀挀攀琀椀挀愀挀椀搀吀愀挀攀琀椀挀愀挀椀搀挀氀愀洀椀氀礀渀栀椀戀
5、椀琀漀爀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀挀愀戀愀搀搀愀愀戀挀攀搀攀昀搀昀搀昀昀挀搀昀昀贀(R)-Filanesib-(R)-ARRY-520)-Kinesin-Inhibitor-MedChemExpress.pdfaaa226879d042c96b67254396caa0cb7d66e0a83d6a904ac3b54086fe555fdff0崁匀漀猀猀礀瀀漀氀愀挀攀琀椀挀愀挀椀搀匀漀猀猀礀瀀漀氀愀挀攀琀椀挀愀挀椀搀挀氀愀洀椀氀礀渀栀椀戀椀琀漀爀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀昀戀昀戀昀搀昀愀挀戀愀挀攀攀搀愀戀搀昀搀愀昀輀(Z)-MDL-105519-MedChemExpress.pdf643031b
6、7ba2781a6aa38bbd74bbe779dbe3a9f1626f41908db3c416ee2e60d490洀圀夀洀吀伀刀渀栀椀戀椀琀漀爀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀挀攀昀攀戀愀愀攀昀戀愀昀搀愀攀昀愀挀搀挀愀搀挀愀鄀kWZ811-CXCR-Antagonist-MedChemExpress.pdf44751a8214923cc08b4caa7cba583daf97f2435ca3ca8b07b0cad17d98521b86s.pdf98d3702ae899b9c0a2c7fd371376afc61e0629d219969481b06da5ba532325010$焀嘀唀洀氀甀刀最漀渀椀猀
7、琀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀挀搀挀昀挀搀搀昀挀昀戀挀戀搀愀昀挀搀昀昀搀攀戀攀挀挀愀挀攀戀蜀qVU-0364439-mGluR-Agonist-MedChemExpress.pdf4334bdaa962da9ad58c792f876106d175031ef8a3746e7f6291d740f98529c070$洀圀夀洀吀伀刀渀栀椀戀椀琀漀爀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀攀攀搀愀愀愀昀攀愀搀戀搀戀攀攀搀搀昀搀攀戀愀搀攀褀WAY-163909-5-HT-Receptor-Agonist-MedChemExpress.pdfffc394026608ed54be59fccb65a37718f662584
8、42a8bb2c47c9130386acb144a0$欀圀倀匀吀吀渀栀椀戀椀琀漀爀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀昀愀昀搀愀愀戀愀愀昀搀戀搀昀戀昀戀攀戀戀挀戀愀攀攀戀謀(R)-(-)-Gossypol-(AT-101)-Bcl-2-Family-Inhibitor-MedChemExpress.pdf22366af51de0a475b8703ed4b39bdde8532b29c2d9d8b14c79cae9d2a5be4bfe0唁刀漀猀猀礀瀀漀氀愀挀攀琀椀挀愀挀椀搀吀愀挀攀琀椀挀愀挀椀搀挀氀愀洀椀氀礀渀栀椀戀椀琀漀爀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀挀愀戀愀搀搀愀愀戀挀攀搀攀昀搀昀搀昀昀挀搀昀昀贀(R)
9、-Filanesib-(R)-ARRY-520)-Kinesin-Inhibitor-MedChemExpress.pdfaaa226879d042c96b67254396caa0cb7d66e0a83d6a904ac3b54086fe555fdff0崁匀漀猀猀礀瀀漀氀愀挀攀琀椀挀愀挀椀搀匀漀猀猀礀瀀漀氀愀挀攀琀椀挀愀挀椀搀挀氀愀洀椀氀礀渀栀椀戀椀琀漀爀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀昀戀昀戀昀搀昀愀挀戀愀挀攀攀搀愀戀搀昀搀愀昀輀(Z)-MDL-105519-MedChemExpress.pdf643031b7ba2781a6aa38bbd74bbe779dbe3a9f1626f41908db3c
10、416ee2e60d490洀圀夀洀吀伀刀渀栀椀戀椀琀漀爀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀挀攀昀攀戀愀愀攀昀戀愀昀搀愀攀昀愀挀搀挀愀搀挀愀:瓄M觜瓄胔-輀K棙齈i缀$Vesnarinone-(OPC-8212)-Phosphodiesterase-(PDE)-Inhibitor-MedChemExpress.pdfpic1.gifVesnarinone(OPC8212)Phosphodiesterase(PDE)InhibitorMedChemExpress.pdf2019-625f9e31fd3-f0f2-41fe-83c5-f7e13234557aotJawxYFzBK17Dnc2V2yObVT
11、YZ5IVDSvacCxHBvVIYhwf5G3xFwXKw=Vesnarinone,OPC,8212,Phosphodiesterase,PDE,Inhibitor,MedChemExpress22b3cec921c855a66c4f0fc2b9e675c0VesnarinoneCat. No.: HY-15297CAS No.: 81840-15-5分式: CHNO分量: 395.45作靶点: Phosphodiesterase (PDE)作通路: Metabolic Enzyme/Protease储存式: Powder -20C 3 years4C 2 yearsIn solvent -
12、80C 6 months-20C 1 month溶解性数据体外实验 DMSO : 16.67 mg/mL (42.15 mM; Need ultrasonic)ConcentrationSolvent Mass 1 mg 5 mg 10 mg1 mM 2.5288 mL 12.6438 mL 25.2876 mL5 mM 0.5058 mL 2.5288 mL 5.0575 mL制备储备液10 mM 0.2529 mL 1.2644 mL 2.5288 mL请根据产品在不同溶剂中的溶解度,选择合适的溶剂配制储备液体内实验 请依序添加每种溶剂: 10% DMSO 40% PEG300 5% Tween-80 45% salineSolubility: 1.67 mg/mL (4.22 mM); Clear solution1. 请依序添加每种溶剂: 10% DMSO 90% corn oilSolubility: 1.67 mg/mL (4.22 mM); Clear solution2. 请依序添加每种溶剂: 10% DMSO 90% (20% SBE-CD in saline)Solubility: 1.67 mg/mL (4.22 mM); Clear solution3. BIOLOGICAL ACTIVITY物活性 Vesnarinone是种喹啉酮衍物, 药效学效应包括