1、OstarineCat. No.: HY-13273CAS No.: 841205-47-8Molecular Formula: CHFNOMolecular Weight: 389.33Target: Androgen ReceptorPathway: OthersStorage: 4C, protect from lightSolvent GTX-024) is a modulator of human androgen receptor.IC50 value:Target: androgen receptorOstarine (MK-2866) is an androgen recept
2、or modulator (SARM) with an ED50 of 0.44 mg/day. Ostarine (MK-2866) has anabolic activity. Lack of PSA increases in men and hair growth in women further corroborated selective anabolic effects of Ostarine (MK-2866). Ostarine (MK-2866) also resulted in a dose-dependent decrease in LDL and HDL cholest
3、erol levels, with the average LDL/HDL ratio for all doses remaining in the low cardiovascular risk catergory.REFERENCES1. Thevis M, et al. Trafficking of drug candidates relevant for sports drug testing: detection of non-approved therapeutics categorized as anabolic and gene doping agents in product
4、s distributed via the Internet.Drug Test Anal. 2011 May;3(5):331-6. doi: 10.1002/dta.283.2. Zilbermint MF, et al. Nonsteroidal selective androgen receptor modulator Ostarine in cancer cachexia. Nonsteroidal selective androgen receptor modulator Ostarine in cancer cachexia.Product Data Sheet InhibitorsAgonistsScreening Librarieswww.MedChemE1Caution: Product has not been fully validated for medical applications. For research use only.Tel: 609-228-6898 Fax: 609-228-5909 E-mail: techMedChemEAddress: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 08852, USAwww.MedChemE2